
RAD-140 (Testolone) is a non-steroidal selective androgen receptor modulator (SARM) designed to exhibit high affinity and specificity for androgen receptors (ARs). It is known for its tissue-selective activity, interacting with androgenic signaling pathways while minimizing off-target interactions. This compound undergoes hepatic metabolism via oxidation and conjugation, with primary clearance occurring through renal and biliary excretion.
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